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Name:LRRK2-IN-1
| Chemical structure | Code NO. |
MT0771 |
 |
Name |
LRRK2-IN-1 |
Synonym |
LRRK 2-IN-1 | |
CAS NO. |
1234480-84-2 | |
Chemical Formula |
C31H38N8O3 | |
MW |
570.69 | |
Purity |
>98% | |
Solubility(R.T.: 25℃) |
100 mM in DMSO; 100 mM in ethanol | |
Stability |
- 20℃, 2 years |
Availability and price
LRRK2-IN-1 is in stock. Bulk available at low price, welcom to inquire quotation.
We offer big discount for bulk quantities. If you have any other questions or needs, please send email to sales@meditechbs.com. We’ll reply you asap.
Description
LRRK2-IN-1 is a cell-permeable, ATP competitive, potent, and selective LRRK2 inhibitor. IC50 is 13 nM, 6 nM, and 2.45 μM for wild type, G2019S mutant, and drug resistant A2016T mutant LRRK2, respectively.
IC50 Value: 13 nM (wild type); 6 nM (G2019S mutant); 2.45 μM (drug resistant A2016T mutant LRRK2)
Target: LRRK2; Mutant LRRK2
LRRK2-IN-1 is useful in treatment of Parkinson's disease.
IC50 Value: 13 nM (wild type); 6 nM (G2019S mutant); 2.45 μM (drug resistant A2016T mutant LRRK2)
Target: LRRK2; Mutant LRRK2
LRRK2-IN-1 is useful in treatment of Parkinson's disease.
References
Attention
Sold for research purposes only; not for human use of any kind.
